Table 2 of Tsai, Mol Vis 2011; 17:1564-1576.


Table 2. Various PKC isozyme inhibitors

Inhibitors PKC isozyme IC50*
Bisindolymaleimide (PKC α, δ, ζ, η, ε) 2–5 μM
Go6976 (PKCα.β.γ) 2–10 nM
Rottlerin (PKCδ) 3–6 μM
HBDDE (PKCα.γ) 43 μM, 50 μM
DAPH-7 (PKCβII.βI) 410 nM, 3.8 μM
Ro32–0432 (PKCα. βI) 9 nM, 28 nM
RBX (PKC βII) 1–2 μM