Table 2 of Tsai, Mol Vis 2011; 17:1564-1576.
Inhibitors | PKC isozyme | IC50* |
---|---|---|
Bisindolymaleimide | (PKC α, δ, ζ, η, ε) | 2–5 μM |
Go6976 | (PKCα.β.γ) | 2–10 nM |
Rottlerin | (PKCδ) | 3–6 μM |
HBDDE | (PKCα.γ) | 43 μM, 50 μM |
DAPH-7 | (PKCβII.βI) | 410 nM, 3.8 μM |
Ro32–0432 | (PKCα. βI) | 9 nM, 28 nM |
RBX | (PKC βII) | 1–2 μM |