Table 4 of Hou, Mol Vis 2010; 16:1659-1668.
Parameters | 10 mg/kg | 25 mg/kg | 50 mg/kg |
---|---|---|---|
Tmax (h) | 0.75±0.27 | 0.58 ±0.20 | 0.50±0.01 |
Cmax (μg/ml) | 24.75±0.85 | 56.77±21.13 | 200.77±32.12 |
t1/2α (h) | 2.15±0.81 | 1.60±0.28 | 0.81±0.60 |
t1/2β (h) | 3.12±0.04 | 1.61±0.31 | 3.25±1.82 |
AUC0-t (μg/ml·h−1) | 121.48±12.92 | 205.28±104.30 | 577.71±63.30 |
K21 (h−1) | 0.09±0.10 | 0.37±0.19 | 0.60±0.57 |
K10 (h−1) | 0.18±0.01 | 0.35±0.05 | 0.58±0.37 |
K12 (h−1) | 0.17±0.10 | 0.22±0.25 | 1.28±1.90 |
MRT0-t (h) | 5.89±0.06 | 4.23±0.66 | 3.10±0.23 |
CL (L/kg·h−1) | 0.06±0.01 | 0.13±0.06 | 0.07 ±0.01 |