Table 1 of Dejneka, Mol Vis 2008; 14:997-1005.


Table 1. Mean concentration of radioactivity in ocular tissues of Dutch-Belted rabbits following a single intravitreal bolus injection of 3H-bevasiranib.




Concentration of radioactivity, μg eq/ga
Group Sex Sample 6 h 24 h 72 h 168 h
1 Males Aqueous fluid 12.3 20.1 11 1.1
1 Males Eye (right) 205 105.1 71.3 18.3
1 Males Iris 12.8 31.7 50 21
1 Males Retina 103.7 221.5 370.2 250.6
1 Males Sclera (+ choroid) 65.4 88.7 54.3 27
1 Males Vitreous fluid 429.3 273.9 118.6 10.4
1 Females Aqueous fluid 3.9 28.9 10.5 1.2
1 Females Eye (right) 175 162 59.4 21.1
1 Females Iris 6.4 37.3 36.4 28.2
1 Females Retina 91 193.8 342.8 278.3
1 Females Sclera (+ choroid) 57 75.6 54.6 24.4
1 Females Vitreous fluid 355.2 307.6 113.7 12.2
2 Males Aqueous fluid 79.8 125.1 90.8 20.2
2 Males Eye (right) 781.2 599.8 483 148.9
2 Males Iris 79.3 134.9 188.6 126.7
2 Males Retina 380.2 416 654.5 682.7
2 Males Sclera (+ choroid) 340.6 329 207.7 100.6
2 Males Vitreous fluid 1919.3 1357.1 777.8 200.7
2 Females Aqueous fluid 119.9 126.9 52.1 19.9
2 Females Eye (right) 818.2 553.9 438.6 159.3
2 Females Iris 139.3 149 92.1 118.7
2 Females Retina 436.1 439.9 449 628.1
2 Females Sclera (+ choroid) 381.1 363 124.7 85.7
2 Females Vitreous fluid 1748.3 1362.6 504.4 205.9